Discovery of allosteric binding sites by crystallographic fragment screening
T. Krojer, James S. Fraser, F. von Delft
Topics & Concepts
Allosteric regulationDrug discoveryComputational biologyFunction (biology)Protein functionFragment (logic)Allosteric enzymeBinding sitePlasma protein bindingChemistryBiologyComputer scienceBioinformaticsBiochemistryGeneticsReceptorGeneProgramming languageComputational Drug Discovery MethodsProtein Structure and DynamicsEnzyme Structure and Function