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Design, synthesis and molecular modeling study of certain quinazolinone derivatives targeting poly (ADP-ribose) polymerase 1 (PARP-1) enzyme as anti-breast cancer and radio-sensitizers

Walid M. Ghorab, Samiha A. El‐Sebaey, Mostafa M. Ghorab

2022Journal of Molecular Structure15 citationsDOI

Topics & Concepts

ChemistryQuinazolinonePoly ADP ribose polymeraseEnzymePolymeraseBreast cancerCombinatorial chemistryCancer researchMolecular modelStereochemistryCancerBiochemistryInternal medicineMedicineBiologyPARP inhibition in cancer therapyToxin Mechanisms and ImmunotoxinsIntegrated Circuits and Semiconductor Failure Analysis
Design, synthesis and molecular modeling study of certain quinazolinone derivatives targeting poly (ADP-ribose) polymerase 1 (PARP-1) enzyme as anti-breast cancer and radio-sensitizers | Litcius