Sensitive fluorogenic substrates for sirtuin deacylase inhibitor discovery
Lingling Yang, Huali Wang, Yu‐Hang Yan, Sha Liu, Zhujun Yu, Meng-Yi Huang, Yubin Luo, Xi Zheng, Yamei Yu, Guo‐Bo Li
Topics & Concepts
ChemistrySirtuinSirtuin 1Drug discoveryPharmacologyStereochemistryBiochemistryEnzymeNAD+ kinaseGeneDownregulation and upregulationMedicineSirtuins and Resveratrol in MedicineAutophagy in Disease and TherapyCancer, Hypoxia, and Metabolism