Valeriaquinone A, a unique anthraquinone–coumarin hybrid with selective inhibition of PTP1B from Knoxia valerianoides
Yan Jiang, Ren‐Yong Yang, Zhao-Xia Qu, Gui‐Ge Hou, Wei Cong, Chunhua Wang, Feng Zhao
Topics & Concepts
CoumarinChemistryAllosteric regulationProtein tyrosine phosphataseStereochemistryAnthraquinoneIC50Docking (animal)SelectivityPhosphataseBiochemistryTyrosineEnzymeIn vitroCatalysisOrganic chemistryNursingMedicineProtein Tyrosine PhosphatasesMorinda citrifolia extract usesBioactive Compounds and Antitumor Agents