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Discovery and optimization of indirubin derivatives as novel ferroptosis inducers for the treatment of colon cancer

Jiangmin Zhu, Chen Chen, Min Kong, Ling Zhu, Yalin Li, Jianfei Zhang, Zhanpeng Yu, Shi-shu Xu, Ling‐Yi Kong, Jian‐Guang Luo, Jian‐Guang Luo

2023European Journal of Medicinal Chemistry16 citationsDOIOpen Access PDF

Topics & Concepts

GPX4ChemistryInducerIn vivoAntioxidantCytotoxicityGlutathioneCancer cellCancer researchEnzymeColorectal cancerCancerBiochemistryPharmacologyGlutathione peroxidaseIn vitroBiologyGeneGeneticsBiotechnologyFerroptosis and cancer prognosisCancer Mechanisms and TherapyPeptidase Inhibition and Analysis
Discovery and optimization of indirubin derivatives as novel ferroptosis inducers for the treatment of colon cancer | Litcius