Imidazo[2,1-b] [1,3,4]thiadiazoles with antiproliferative activity against primary and gemcitabine-resistant pancreatic cancer cells
Stella Cascioferro, Giovanna Li Petri, Barbara Parrino, Daniela Carbone, Niccola Funel, Cecilia Bergonzini, Giulia Mantini, Henk Dekker, Daan P. Geerke, Godefridus J. Peters, Girolamo Cirrincione, Elisa Giovannetti, Patrizia Diana
Topics & Concepts
ChemistryPancreatic cancerGemcitabineCancer researchCell cultureIC50Focal adhesionKinaseIn vitroPhosphorylationMolecular biologyBiochemistryCancerInternal medicineBiologyGeneticsMedicineQuinazolinone synthesis and applicationsSynthesis and biological activityCancer Mechanisms and Therapy