Asymmetric drug binding in an ATP-loaded inward-facing state of an ABC transporter
Tarjani Thaker, Smriti Mishra, Wenchang Zhou, Michael J. Mohan, Qingyu Tang, José D. Faraldo‐Gómez, Hassane S. Mchaourab, Thomas Tomasiak
Topics & Concepts
ATP-binding cassette transporterFlippaseTransmembrane domainBiophysicsATP hydrolysisCyclic nucleotide-binding domainTransporterEffluxBinding siteElectron transport chainChemistrySubstrate (aquarium)Adenosine triphosphateProtein structureBiochemistryNucleotideBiologyATPaseEnzymeMembranePhospholipidGenePhosphatidylserineEcologyDrug Transport and Resistance MechanismsTrace Elements in HealthDNA and Nucleic Acid Chemistry