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Fused chromeno and quinolino[1,8]naphthyridines: Synthesis and biological evaluation as topoisomerase I inhibitors and antiproliferative agents

Endika Martín‐Encinas, Gloria Rubiales, Birgitta R. Knudsen, Francisco Palácios, Concepción Alonso

2021Bioorganic & Medicinal Chemistry20 citationsDOI

Topics & Concepts

ChemistryCamptothecinTopoisomeraseStereochemistryCombinatorial chemistryCycloadditionCell cultureEnzymeOrganic chemistryCatalysisBiologyGeneticsCancer therapeutics and mechanismsBioactive Compounds and Antitumor AgentsSynthesis and biological activity
Fused chromeno and quinolino[1,8]naphthyridines: Synthesis and biological evaluation as topoisomerase I inhibitors and antiproliferative agents | Litcius