Discovery of Thai mangrove tetranortriterpenoids as agonists of human pregnane–X–receptor and inhibitors against human carboxylesterase 2
Yan-Xia Ren, Xiaopeng Zou, Wan‐Shan Li, Jun Wu, Li Shen
Topics & Concepts
ChemistryStereochemistryPregnane X receptorCarboxylesteraseElectrospray ionizationCircular dichroismPharmacologyBiochemistryEnzymeMass spectrometryChromatographyGeneNuclear receptorMedicineTranscription factorPhytochemical compounds biological activitiesTraditional and Medicinal Uses of AnnonaceaeMarine Sponges and Natural Products