Discovery of tertiary amide derivatives incorporating benzothiazole moiety as anti-gastric cancer agents in vitro via inhibiting tubulin polymerization and activating the Hippo signaling pathway
Jian Song, Qiu-Lei Gao, Bowen Wu, Ting Zhu, Xinxin Cui, Chengjun Jin, Shuyu Wang, Shenghui Wang, Dong‐Jun Fu, Hong‐Min Liu, Sai‐Yang Zhang, Yanbing Zhang, Yongchun Li
Topics & Concepts
ChemistryTubulinBenzothiazoleIn vitroHippo signaling pathwayCancer cellDocking (animal)MicrotubuleCell growthStereochemistryCell biologyBiochemistryCancerBiologyNursingGeneticsMedicineHippo pathway signaling and YAP/TAZPI3K/AKT/mTOR signaling in cancer14-3-3 protein interactions