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Improved l-Type amino acid transporter 1 (LAT1)-mediated delivery of anti-inflammatory drugs into astrocytes and microglia with reduced prostaglandin production

Janne Tampio, Susanne Löffler, Melina Guillon, Agathe Hugele, Johanna Huttunen, Kristiina M. Huttunen

2021International Journal of Pharmaceutics26 citationsDOI

Topics & Concepts

MicrogliaProdrugPharmacologyKetoprofenChemistryViability assayIbuprofenProstaglandin E2Blood–brain barrierNaproxenInflammationProstaglandinLipopolysaccharideBiochemistryCellMedicineImmunologyCentral nervous systemInternal medicinePathologyAlternative medicineAmino Acid Enzymes and MetabolismNeuroscience and Neuropharmacology ResearchDrug Transport and Resistance Mechanisms
Improved l-Type amino acid transporter 1 (LAT1)-mediated delivery of anti-inflammatory drugs into astrocytes and microglia with reduced prostaglandin production | Litcius