Litcius/Paper detail

Analysis of lorlatinib analogs reveals a roadmap for targeting diverse compound resistance mutations in ALK-positive lung cancer

Aya Shiba‐Ishii, Ted W. Johnson, Ibiayi Dagogo‐Jack, Mari Mino–Kenudson, Theodore R. Johnson, Ping Wei, Scott L. Weinrich, Michele McTigue, Makeba Walcott, Linh Nguyen-Phuong, Kristin Dionne, Adam Acker, Lesli A. Kiedrowski, Andrew Do, Jennifer Peterson, Jaimie L. Barth, Beow Y. Yeap, Justin F. Gainor, Jessica J. Lin, Satoshi Yoda, Aaron N. Hata

2022Nature Cancer69 citationsDOIOpen Access PDF

Topics & Concepts

Anaplastic lymphoma kinaseALK inhibitorCancer researchTyrosine kinaseTyrosine-kinase inhibitorLung cancerMutantKinaseMutationAcquired resistanceTargeted therapyBiologyCancerPharmacologyGeneGeneticsMedicineSignal transductionInternal medicineMalignant pleural effusionLung Cancer Treatments and MutationsCancer therapeutics and mechanismsLung Cancer Research Studies
Analysis of lorlatinib analogs reveals a roadmap for targeting diverse compound resistance mutations in ALK-positive lung cancer | Litcius