Litcius/Paper detail

Activation and Signaling Mechanism Revealed by Cannabinoid Receptor-Gi Complex Structures

Tian Hua, Xiaoting Li, Lijie Wu, Christos Iliopoulos‐Tsoutsouvas, Yuxia Wang, Meng Wu, Ling Shen, Christina A. Brust, Spyros P. Nikas, Feng Song, Xiyong Song, Shuguang Yuan, Qianqian Sun, Yiran Wu, Shan Jiang, Travis W. Grim, Othman Benchama, Edward L. Stahl, Nikolai Zvonok, Suwen Zhao, Laura Bohn, Alexandros Makriyannis, Zhi‐Jie Liu

2020Cell352 citationsDOIOpen Access PDF

Topics & Concepts

Cannabinoid receptorAgonistBiologyEndocannabinoid systemCannabinoidAllosteric regulationMechanism (biology)G protein-coupled receptorInverse agonistCannabinoid receptor type 2ReceptorSignal transductionNeuroscienceDrug discoveryCell biologyPharmacologyBiochemistryEpistemologyPhilosophyCannabis and Cannabinoid ResearchPharmacological Receptor Mechanisms and EffectsNeuroscience and Neuropharmacology Research