Novel Potent Muscarinic Receptor Antagonists: Investigation on the Nature of Lipophilic Substituents in the 5- and/or 6-Positions of the 1,4-Dioxane Nucleus
Fabio Del Bello, Alessandro Bonifazi, Gianfabio Giorgioni, Alessandro Piergentili, Maria Giovanna Sabbieti, Dimitrios Agas, Marzia Dell’Aera, Rosanna Matucci, Marcin Górecki, Gennaro Pescitelli, Giulio Vistoli, Wilma Quaglia
Abstract
receptors are involved.
Topics & Concepts
ChemistryMuscarinic acetylcholine receptorMoietyStereochemistrySelectivityAntagonistDocking (animal)EnantiomerReceptorBiochemistryMedicineNursingCatalysisReceptor Mechanisms and SignalingCardiac electrophysiology and arrhythmiasIon channel regulation and function