Discovery of a novel water-soluble, rapid-release triptolide prodrug with improved drug-like properties and high efficacy in human acute myeloid leukemia
Di Kang, Xiang Pan, Yi Song, Yan Liu, Dan Wang, Xuejun Zhu, Junwei Wang, Lihong Hu
Topics & Concepts
TriptolideProdrugChemistryMyeloid leukemiaPharmacologyPharmacokineticsLinkerDrugBiochemistryCancer researchMedicineApoptosisOperating systemComputer scienceNatural Compounds in Disease TreatmentHistone Deacetylase Inhibitors ResearchAcute Myeloid Leukemia Research