Industry Perspective on the Pharmacokinetic and Absorption, Distribution, Metabolism, and Excretion Characterization of Heterobifunctional Protein Degraders
Laurie P. Volak, Heide Marika Duevel, Sara C. Humphreys, David O. Nettleton, Colin Phipps, Andy Pike, Caroline Rynn, Paul Scott‐Stevens, Donglu Zhang, Michael Zientek
Topics & Concepts
ADMELipinski's rule of fiveBioavailabilityPharmacokineticsIn silicoChemistryComputational biologyDNA ligasePharmacologyBiochemistryBiochemical engineeringBiologyEngineeringEnzymeGeneProtein Degradation and InhibitorsProtein purification and stabilitySoftware Testing and Debugging Techniques