Design, synthesis, and bioactivity evaluation of novel amide/sulfonamide derivatives as potential anti-inflammatory agents against acute lung injury and ulcerative colitis
Pan Chen, Jun Yang, Ying Zhou, Xiaobo Li, Yu Zou, Zhiwei Zheng, Mi Guo, Zhichao Chen, Won‐Jea Cho, Nipon Chattipakorn, Wenqi Wu, Qidong Tang, Guang Liang
Topics & Concepts
Ulcerative colitisChemistrySulfonamideAmideIn vivoPharmacologyInflammationAnti-inflammatoryTumor necrosis factor alphaProinflammatory cytokineIC50Inflammatory bowel diseaseIn vitroColitisBiochemistryStereochemistryImmunologyMedicineInternal medicineBiologyBiotechnologyDiseaseQuinazolinone synthesis and applicationsSynthesis and biological activityPneumocystis jirovecii pneumonia detection and treatment