Structural identification of lysophosphatidylcholines as activating ligands for orphan receptor GPR119
Peiyu Xu, Sijie Huang, Shimeng Guo, Ying Yun, Xi Cheng, Xinheng He, Pengjun Cai, Yuan Lan, Hu Zhou, Hualiang Jiang, Yi Jiang, Xin Xie, H. Eric Xu
Topics & Concepts
G protein-coupled receptorReceptorLysophosphatidylcholineOrphan receptorBiochemistryChemistryCell biologyBiologyPhosphatidylcholinePhospholipidMembraneTranscription factorGeneReceptor Mechanisms and SignalingSphingolipid Metabolism and SignalingDiabetes Treatment and Management