Anti-inflammatory efficacy and relevant SAR investigations of novel chiral pyrazolo isoquinoline derivatives: Design, synthesis, in-vitro, in-vivo, and computational studies targeting iNOS
Maryam Akhtar, Jiabin Niu, Yujie Zhu, Zhaoyi Luo, Ting Tian, Yuanliang Dong, Yuan Wang, Muhammad Subaan Fareed, Li Lin
Topics & Concepts
ChemistryIsoquinolineIn vivoIn vitroStereochemistryPharmacologyCombinatorial chemistryBiochemistryBiotechnologyMedicineBiologySynthesis and biological activityComputational Drug Discovery MethodsSynthesis of heterocyclic compounds