A dual-acting 5-HT6 receptor inverse agonist/MAO-B inhibitor displays glioprotective and pro-cognitive properties
Vittorio Canale, Katarzyna Grychowska, Rafał Kurczab, Mateusz Ryng, Abdul Raheem Keeri, Grzegorz Satała, Agnieszka Olejarz‐Maciej, Paulina Koczurkiewicz, Marcin Drop, Klaudia Blicharz, Kamil Piska, Elżbieta Pękala, Paulina Janiszewska, Martyna Krawczyk, Maria Walczak, Séverine Chaumont‐Dubel, Andrzej J. Bojarski, Philippe Marin, Piotr Popik, Paweł Zajdel
Topics & Concepts
Inverse agonistChemistryPharmacophore5-HT6 receptorPharmacologyAgonistReceptorContext (archaeology)NeuroscienceStereochemistryBiochemistryPsychology5-HT receptorSerotoninMedicineBiologyPaleontologyPhosphodiesterase function and regulationReceptor Mechanisms and SignalingNeuroscience and Neuropharmacology Research