Design, synthesis and bioactivity study on 5-phenylfuran derivatives as potent reversal agents against P-glycoprotein-mediated multidrug resistance in MCF-7/ADR cell
Yasheng Li, Xi Yang, Dongsheng Zhao, Yue Cai, Zhi Huang, Rui Wu, Sijia Wang, Guijun Liu, Jian Wang, Xiaoze Bao, Xinyi Ye, Bin Wei, Zi‐Ning Cui, Hong Wang
Topics & Concepts
P-glycoproteinMultiple drug resistanceChemistryDoxorubicinEffluxPharmacologyVincristineDrug resistanceIC50PaclitaxelIn vitroBiochemistryChemotherapyMedicineBiologyInternal medicineCyclophosphamideMicrobiologyAntibioticsDrug Transport and Resistance MechanismsCancer therapeutics and mechanismsHIV/AIDS drug development and treatment