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Molecular mechanisms of AMPK/YAP/NLRP3 signaling pathway affecting the occurrence and development of ankylosing spondylitis

Ruiyang Fu, Xiaoqing Guo, Zhongqiang Pan, Yaling Wang, Jing Xu, Lei Zhang, Jinxia Li

2023Journal of Orthopaedic Surgery and Research17 citationsDOIOpen Access PDF

Abstract

BACKGROUND: Investigate the AMPK (protein kinase AMP-activated catalytic subunit alpha 1)/YAP (Yes1 associated transcriptional regulator)/NLRP3 (NLR family pyrin domain containing 3) signaling pathway's role in ankylosing spondylitis (AS) development using public database analysis, in vitro and in vivo experiments. METHODS: Retrieve AS dataset, analyze differential gene expression in R, conduct functional enrichment analysis, collect 30 AS patient and 30 normal control samples, and construct a mouse model. ELISA, IP, and knockdown experiments were performed to detect expression changes. RESULTS: NLRP3 was identified as a significant AS-related gene. Caspase-1, IL-1β, IL-17A, IL-18, IL-23, YAP, and NLRP3 were upregulated in AS patients. Overexpressing AMPK inhibited YAP's blockade on NLRP3 ubiquitination, reducing ossification in fibroblasts. Inhibiting AMPK exacerbated AS symptoms in AS mice. CONCLUSION: AMPK may suppress YAP expression, leading to NLRP3 inflammasome inhibition and AS alleviation.

Topics & Concepts

AMPKMedicineGene knockdownInflammasomePyrin domainDownregulation and upregulationAnkylosing spondylitisSignal transductionRegulatorProtein kinase ACell biologyCancer researchKinaseImmunologyGeneBiologyInflammationGeneticsSpondyloarthritis Studies and TreatmentsInflammasome and immune disordersOsteomyelitis and Bone Disorders Research