Tailored horseshoe-shaped nicotinonitrile scaffold as dual promising c-Met and Pim-1 inhibitors: Design, synthesis, SAR and in silico study
Samy Mohamady, Ahmed Khalil, Bassem H. Naguib, Mohamed S. Nafie, Haytham O. Tawfik, Moataz A. Shaldam
Topics & Concepts
ChemistryKinaseMTT assayCytotoxicityCell cultureIC50In silicoApoptosisBiochemistryIn vitroStereochemistryBiologyGeneGeneticsCancer Mechanisms and TherapySynthesis and biological activitySynthesis and bioactivity of alkaloids