Structural Insights into the Catalytic Cycle of a Bacterial Multidrug ABC Efflux Pump
Waqas Javed, Sylvain D. Vallet, Marie-Pierre Clement, Aline Le Roy, Martine Moulin, Michael Härtlein, Cécile Breyton, Odile Burlet‐Schiltz, Julien Marcoux, Cédric Orelle, Christine Ebel, Anne Martel, Jean‐Michel Jault
Topics & Concepts
ATP-binding cassette transporterEffluxSubfamilyVanadateATPaseTransporterChemistryATP hydrolysisBiochemistryCatalytic cycleStereochemistryBiologyEnzymeGeneDrug Transport and Resistance MechanismsAntibiotic Resistance in BacteriaAntibiotics Pharmacokinetics and Efficacy