Litcius/Paper detail

Accurately Predicting Protein p <i>K</i> <sub>a</sub> Values Using Nonequilibrium Alchemy

Carter J. Wilson, Mikko Karttunen, Bert L. de Groot, Vytautas Gapsys

2023Journal of Chemical Theory and Computation22 citationsDOIOpen Access PDF

Abstract

values of coupled residues and observe a substantial performance disparity associated with the lysine partial charges in Amber14SB/Amber99SB*-ILDN, for which an underused fix already exists.

Topics & Concepts

ProtonationNon-equilibrium thermodynamicsChemistryThermodynamicsStatistical physicsLysinePhysicsComputational chemistryBiological systemAmino acidIonBiochemistryOrganic chemistryBiologyComputational Drug Discovery MethodsProtein Structure and DynamicsFree Radicals and Antioxidants
Accurately Predicting Protein p <i>K</i> <sub>a</sub> Values Using Nonequilibrium Alchemy | Litcius