Mechanism of gating and partial agonist action in the glycine receptor
Jie Yu, Hongtao Zhu, Remigijus Lapė, Timo Greiner, Juan Du, Wei Lü, Lucia G. Sivilotti, Eric Gouaux
Topics & Concepts
Partial agonistAgonistBiologyBiophysicsGlycine receptorReceptorNeurotransmitter receptorIntrinsic activityNeurotransmitterIon channelLigand-gated ion channelSignal transductionBiochemistryCell biologyGlycineAmino acidNicotinic Acetylcholine Receptors StudyIon channel regulation and functionReceptor Mechanisms and Signaling