Activation loop phosphorylation tunes conformational dynamics underlying Pyk2 tyrosine kinase activation
Tânia Marina Palhano Zanela, Alexzandrea Woudenberg, Karen G. Romero Bello, Eric S. Underbakke
Topics & Concepts
AutophosphorylationProto-oncogene tyrosine-protein kinase SrcPhosphorylationFERM domainCell biologyChemistryProtein kinase domainBiophysicsBiochemistryBiologyProtein kinase AMutantGeneMembrane proteinIntegral membrane proteinMembraneProtein Kinase Regulation and GTPase SignalingProtein Structure and DynamicsEnzyme Structure and Function