Litcius/Paper detail

In Situ Alkyl Radical Recycling-Driven Decoupled Electrophotochemical Deamination

Kui Wang, Xiaoyu Liu, Siyu Yang, Yan Tian, Mingyang Zhou, Jianhua Zhou, Xiaofei Jia, Baoying Li, Siyuan Liu, Jianbin Chen

2022Organic Letters47 citationsDOI

Abstract

Molecular electrophotocatalysis has emerged as a powerful strategy for the development of sustainable synthetic protocols. With the proof-of-concept, we exploited a versatile electrophotocatalytic deaminative alkylation approach. Mechanistic investigation indicated that in situ recycling of the alkyl radicals was the key point. Notably, ligand modification and late-stage functionalization of pharmaceuticals were also established, highlighting its feasibility in practical utilization.

Topics & Concepts

ChemistryDeaminationAlkylAlkylationCombinatorial chemistryRadicalIn situSurface modificationOrganic chemistryCatalysisPhysical chemistryEnzymeRadical Photochemical ReactionsCatalytic C–H Functionalization MethodsSulfur-Based Synthesis Techniques