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Benzoxepinones: A new isoform-selective class of tumor associated carbonic anhydrase inhibitors

Aiga Grandāne, Alessio Nocentini, Thomas Werner, Raivis Žalubovskis, Claudiu T. Supuran

2020Bioorganic & Medicinal Chemistry26 citationsDOIOpen Access PDF

Topics & Concepts

Gene isoformChemistryCarbonic anhydraseCytosolIsozymeEnzymeBiochemistryEnzyme inhibitorCarbonic anhydrase IIGeneEnzyme function and inhibitionSynthesis and Catalytic ReactionsChemical Reactions and Mechanisms
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