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Structure-based design of bitopic ligands for the µ-opioid receptor

Abdelfattah Faouzi, Haoqing Wang, Saheem A. Zaidi, Jeffrey F. DiBerto, Tao Che, Qianhui Qu, Michael J. Robertson, Manish K. Madasu, Amal El Daibani, Balázs R. Varga, Tiffany Zhang, Claudia Ruiz, Shan Liu, Jin Xu, Kevin Appourchaux, Samuel T. Slocum, Shainnel O. Eans, Michael D. Cameron, Ream Al‐Hasani, Ying‐Xian Pan, Bryan L. Roth, Jay P. McLaughlin, Georgios Skiniotis, Vsevolod Katritch, Brian K. Kobilka, Susruta Majumdar

2022Nature128 citationsDOIOpen Access PDF

Topics & Concepts

ReceptorChemistryOpioidPharmacologyBinding siteAllosteric regulationFentanylStereochemistryBiochemistryBiologyReceptor Mechanisms and SignalingNeuropeptides and Animal PhysiologyPharmacological Receptor Mechanisms and Effects
Structure-based design of bitopic ligands for the µ-opioid receptor | Litcius