A comparative study on in vitro and in vivo characteristics of enzalutamide nanocrystals versus amorphous solid dispersions and a better prediction for bioavailability based on “spring-parachute” model
Xueting Guo, Yibin Guo, Maolian Zhang, Bing Yang, Hao Liu, Tian Yin, Yu Zhang, Haibing He, Yanjiao Wang, Dongchun Liu, Jingxin Gou, Xing Tang
Topics & Concepts
Amorphous solidMaterials scienceSupersaturationBioavailabilityDissolutionDissolution testingNanocrystalChemical engineeringChromatographyAnalytical Chemistry (journal)NanotechnologyChemistryPharmacologyCrystallographyOrganic chemistryMedicineEngineeringBiopharmaceutics Classification SystemDrug Solubulity and Delivery SystemsCrystallization and Solubility StudiesAdvanced Drug Delivery Systems