Litcius/Paper detail

Design, synthesis, and biological evaluation of novel (4-(1,2,4-oxadiazol-5-yl)phenyl)-2-aminoacetamide derivatives as multifunctional agents for the treatment of Alzheimer's disease

Tongtong Liu, Shiming Chen, Jiyu Du, Siqi Xing, Rong Li, Zeng Li

2021European Journal of Medicinal Chemistry38 citationsDOIOpen Access PDF

Topics & Concepts

ChemistryButyrylcholinesteraseNeuroprotectionPotencyIC50NeuroinflammationLead compoundPharmacologyDPPHReactive oxygen speciesAntioxidantStereochemistryBiochemistryIn vitroInflammationAchéAcetylcholinesteraseEnzymeImmunologyMedicineBiologyCholinesterase and Neurodegenerative DiseasesComputational Drug Discovery MethodsAlzheimer's disease research and treatments