Litcius/Paper detail

Hydroxamic acid hybrids: Histone deacetylase inhibitors with anticancer therapeutic potency

Yuan Jiang Pan, Haodong Hou, Bo Zhou, Jingyue Gao, Feng Gao, Feng Gao

2023European Journal of Medicinal Chemistry24 citationsDOIOpen Access PDF

Topics & Concepts

Histone deacetylaseHydroxamic acidChemistryVorinostatHistonePharmacophoreCell cycle checkpointRational designHistone deacetylase inhibitorSmall moleculeAcetylationCancer researchPharmacologyBiochemistryCell cycleApoptosisBiologyGeneGeneticsStereochemistryHistone Deacetylase Inhibitors ResearchProtein Degradation and InhibitorsPeptidase Inhibition and Analysis