Discovery and development of 2-aminobenzimidazoles as potent antimalarials
Shane M. Devine, Matthew Challis, Jomo K. Kigotho, Ghizal Siddiqui, Amanda De Paoli, Christopher A. MacRaild, Vicky M. Avery, Darren J. Creek, Raymond S. Norton, Peter J. Scammells
Topics & Concepts
Plasmodium falciparumChemistryPharmacophoreMoietyCytotoxicityArtemisininIn vitroPotencyIC50StereochemistryPharmacologyDrug discoveryCombinatorial chemistryBiochemistryMalariaBiologyImmunologyMalaria Research and ControlHIV/AIDS drug development and treatmentComputational Drug Discovery Methods