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Discovery of novel N-sulfonamide-tetrahydroisoquinolines as potent retinoic acid receptor-related orphan receptor γt agonists

Xiaojun Ma, Nannan Sun, Xinwei Li, Wei Fu

2021European Journal of Medicinal Chemistry25 citationsDOIOpen Access PDF

Topics & Concepts

Orphan receptorChemistryRAR-related orphan receptor gammaRetinoic acid receptorAgonistRetinoic acidReceptorNuclear receptorCancer researchPharmacologyTranscription factorStereochemistryBiochemistryGeneBiologyPsoriasis: Treatment and PathogenesisGenomics, phytochemicals, and oxidative stressImmune Cell Function and Interaction
Discovery of novel N-sulfonamide-tetrahydroisoquinolines as potent retinoic acid receptor-related orphan receptor γt agonists | Litcius