Litcius/Paper detail

Physiologically Based Absorption Modelling to Explore the Impact of Food and Gastric pH Changes on the Pharmacokinetics of Entrectinib

Neil Parrott, Cordula Stillhart, Marc Lindenberg, Bjoern Wagner, Karey Kowalski, Elena Guerini, Nassim Djebli, Georgina Meneses‐Lorente

2020The AAPS Journal50 citationsDOI

Topics & Concepts

Physiologically based pharmacokinetic modellingIn silicoPharmacokineticsChemistryPharmacologyBioavailabilityADMEDrugIn vivoDrug developmentBiochemistryMedicineBiotechnologyBiologyGeneDrug Solubulity and Delivery SystemsProtein purification and stabilityDrug Transport and Resistance Mechanisms