Litcius/Paper detail

Simple Synthesis of Amides via Their Acid Chlorides in Aqueous TPGS-750-M

Min Shi, Ning Ye, Wei Chen, Hui Wang, Chi‐Ming Cheung, Michaël Parmentier, Fabrice Gallou, Bin Wu

2020Organic Process Research & Development41 citationsDOI

Abstract

The technology of surfactant chemistry is employed for amide bond construction via the reaction of acyl chlorides with amines in 2 wt % TPGS-750-M aqueous solution. Specifically, this highly efficient method enables a chromatography-free scalable process and recycling of the TPGS-750-M solution.

Topics & Concepts

Aqueous solutionChemistryAmidePulmonary surfactantCombinatorial chemistryOrganic chemistryChromatographyBiochemistryChemical Synthesis and AnalysisChemical Synthesis and ReactionsAnalytical Chemistry and Chromatography