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Metabolism of Speciociliatine, an Overlooked Kratom Alkaloid for its Potential Pharmacological Effects

Shyam H. Kamble, Erin C. Berthold, Siva Rama Raju Kanumuri, Tamara I. King, Michelle A. Kuntz, Francisco León, Marco Mottinelli, Lance Richard McMahon, Christopher R. McCurdy, Abhisheak Sharma

2022The AAPS Journal25 citationsDOIOpen Access PDF

Topics & Concepts

AlkaloidMicrosomeMetabolismPharmacologyCYP3A4Indole alkaloidDemethylationBiologyChemistryIn vitroBiochemistryCytochrome P450StereochemistryGeneGene expressionDNA methylationAlkaloids: synthesis and pharmacologyTraditional and Medicinal Uses of AnnonaceaeBerberine and alkaloids research
Metabolism of Speciociliatine, an Overlooked Kratom Alkaloid for its Potential Pharmacological Effects | Litcius