Design, synthesis, antitumor activity and theoretical calculation of novel PI3Ka inhibitors
Ruyi Jin, Tian Tang, Sha Zhou, Long Xu, Hui Guo, Jing Zhou, Hao Yan, Zhi Li, Zheng‐Yu Zuo, Honglei Xie, Yuping Tang
Topics & Concepts
ChemistryThiazoleSelectivityCombinatorial chemistryAutoDockStereochemistryPurineHOMO/LUMODrugEnzymeBiochemistryPharmacologyGeneOrganic chemistryMoleculeIn silicoCatalysisMedicinePI3K/AKT/mTOR signaling in cancerChronic Lymphocytic Leukemia ResearchProtein Degradation and Inhibitors