Development of BRD4 inhibitors as anti-inflammatory agents and antidotes for arsenicals
Marina Fosso Yatchang, Bini Mathew, Ritesh K. Srivastava, Jasim Khan, Suhail Muzaffar, Sixue Zhang, Mousheng Wu, Ling Zhai, Pedro Ruiz, Anupam Agarwal, J. Robert Bostwick, Mark J. Suto, Mohammad Athar, Corinne E. Augelli‐Szafran
Topics & Concepts
BromodomainChemistryBRD4Context (archaeology)PharmacologySmall moleculeDrug discoveryBiochemistryEpigeneticsMedicineBiologyGenePaleontologyProtein Degradation and InhibitorsMultiple Myeloma Research and TreatmentsAdvanced biosensing and bioanalysis techniques