Development of triazolothiadiazine derivatives as highly potent tubulin polymerization inhibitors: Structure-activity relationship, in vitro and in vivo study
Weifeng Ma, Peng Chen, Xian‐Sen Huo, Yufeng Ma, Yanhong Li, Peng-Cheng Diao, Fang Yang, Shengquan Zheng, Meng‐Jin Hu, Wen‐Wei You, Pei‐Liang Zhao
Topics & Concepts
ChemistryIn vivoIn vitroCyclin B1ApoptosisTubulinCyclin-dependent kinase 1Cell cycleCell growthCell cycle checkpointMicrotubule polymerizationMicrotubuleBiochemistryCell biologyBiologyBiotechnologySynthesis and biological activityClick Chemistry and ApplicationsQuinazolinone synthesis and applications