A novel class of selective CK2 inhibitors targeting its open hinge conformation
Andrea Dalle Vedove, Francesca Zonta, Enrico Zanforlin, Nicola Demitri, Giovanni Ribaudo, Giulia Cazzanelli, Alberto Ongaro, Stefania Sarno, Giuseppe Zagotto, Roberto Battistutta, Maria Ruzzene, Graziano Lolli
Topics & Concepts
ChemistryKinaseStereochemistrySelectivityRing (chemistry)BiochemistryCombinatorial chemistryCatalysisOrganic chemistryProtein Kinase Regulation and GTPase SignalingUbiquitin and proteasome pathwaysBiochemical and Molecular Research