Novel quinoline-based derivatives: A new class of PDE4B inhibitors for adjuvant-induced arthritis
Siqi Xing, Weizheng Fan, Junhua Chen, Jiyu Du, Tongtong Liu, Shuanghong Dong, Jucheng Xia, Peipei Liu, Dexing Zou, Cai Li, Zeng Li
Topics & Concepts
ChemistryPharmacologyIC50Western blotIn vivoArthritisLipopolysaccharideQuinolineIn vitroInflammationTumor necrosis factor alphaProinflammatory cytokineBiochemistryImmunologyMedicineBiologyOrganic chemistryBiotechnologyGenePhosphodiesterase function and regulationPhenothiazines and Benzothiazines Synthesis and ActivitiesSynthesis and biological activity