Selective degradation of BRD4 suppresses lung cancer cell proliferation using GSH-responsive PROTAC precursors
Heli Fan, Zhili Zhou, Dehao Yu, Jing Sun, Luo Wang, Yuanyuan Jia, Junyu Tian, Wenyi Mi, Huabing Sun, Huabing Sun
Topics & Concepts
ChemistryGlutathioneCancer cellProteasomeCancerCancer researchProtein degradationProteolysisLung cancerCell growthBRD4Cell biologyIntracellularEpigeneticsPharmacologyBiochemistryBiologyMedicineInternal medicineBromodomainEnzymeGeneProtein Degradation and InhibitorsUbiquitin and proteasome pathwaysMultiple Myeloma Research and Treatments