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Inhibition of human UDP-glucuronosyltransferase enzyme by ripretinib: Implications for drug-drug interactions

Xin Lv, Zhe Wang, Zhen Wang, Hang Yin, Yangliu Xia, Lili Jiang, Yong Liu

2023Toxicology and Applied Pharmacology11 citationsDOI

Topics & Concepts

PharmacologyEnzymeDrugIn vivoChemistryIC50In vitroMedicineBiochemistryBiologyBiotechnologyPI3K/AKT/mTOR signaling in cancerPharmacogenetics and Drug MetabolismChronic Lymphocytic Leukemia Research
Inhibition of human UDP-glucuronosyltransferase enzyme by ripretinib: Implications for drug-drug interactions | Litcius