Litcius/Paper detail

Discovery of methoxy-naphthyl linked N-(1-benzylpiperidine) benzamide as a blood-brain permeable dual inhibitor of acetylcholinesterase and butyrylcholinesterase

Mohd Abdullaha, Vijay K. Nuthakki, Sandip B. Bharate

2020European Journal of Medicinal Chemistry34 citationsDOIOpen Access PDF

Topics & Concepts

ButyrylcholinesteraseChemistryAcetylcholinesteraseBenzamideCholinesteraseAcetylcholinePharmacologyAchéStereochemistryDocking (animal)NeurotransmissionEnzymeBiochemistryReceptorNursingMedicineCholinesterase and Neurodegenerative DiseasesComputational Drug Discovery MethodsPesticide Exposure and Toxicity