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Celastrol as an intestinal FXR inhibitor triggers tripolide-induced intestinal bleeding: Underlying mechanism of gastrointestinal injury induced by Tripterygium wilfordii

Manyun Dai, Wan Peng, Lisha Lin, Zhanxuan E. Wu, Ting Zhang, Qi Zhao, Yan Cheng, Qiuxia Lin, Binbin Zhang, Aiming Liu, Qianru Rao, Jian‐Feng Huang, Jinhua Zhao, Frank J. Gonzalez, Fei Li, Fei Li

2023Phytomedicine19 citationsDOI

Topics & Concepts

CelastrolTriptolideTripterygium wilfordiiTripterygiumFarnesoid X receptorPharmacologyChemistryDownregulation and upregulationApoptosisMedicineBiochemistryNuclear receptorPathologyTranscription factorGlycosideGeneAlternative medicineOrganic chemistryNatural Compounds in Disease TreatmentInflammatory Bowel DiseaseLiver physiology and pathology
Celastrol as an intestinal FXR inhibitor triggers tripolide-induced intestinal bleeding: Underlying mechanism of gastrointestinal injury induced by Tripterygium wilfordii | Litcius