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Hyperactivation of TORC1 Drives Resistance to the Pan-HER Tyrosine Kinase Inhibitor Neratinib in HER2-Mutant Cancers

Dhivya R. Sudhan, Ángel Guerrero‐Zotano, Helen Won, Paula González Ericsson, Alberto Servetto, Mariela Huerta-Rosario, Dan Ye, Kyung‐min Lee, Luigi Formisano, Yan Guo, Qi Liu, Lisa N. Kinch, Monica Red Brewer, Teresa C. Dugger, James P. Koch, Michael J. Wick, Richard E. Cutler, Alshad S. Lalani, Richard Bryce, Alan Auerbach, Ariella B. Hanker, Carlos L. Arteaga

2020Cancer Cell49 citationsDOIOpen Access PDF

Topics & Concepts

NeratinibCancer researchBiologyTyrosine-kinase inhibitorCancerGeneticsBreast cancerTrastuzumabPI3K/AKT/mTOR signaling in cancerHER2/EGFR in Cancer ResearchChronic Lymphocytic Leukemia Research
Hyperactivation of TORC1 Drives Resistance to the Pan-HER Tyrosine Kinase Inhibitor Neratinib in HER2-Mutant Cancers | Litcius