Pharmacological characterization of novel synthetic opioids: Isotonitazene, metonitazene, and piperidylthiambutene as potent μ-opioid receptor agonists
Maria Antonietta De Luca, Graziella Tocco, Rafaela Mostallino, Antonio Laus, Francesca Caria, Aurora Musa, Nicholas Pintori, Marcos Ucha, Celia Poza, Emilio Ambrosio, G. Di Chiara, M. Paola Castelli
Topics & Concepts
DAMGOChemistryPotencyPharmacologyOpioidMorphineOpioid receptorED50AgonistFentanylIntrinsic activityEnkephalinReceptorIn vitroBiochemistryMedicineReceptor Mechanisms and SignalingNeuropeptides and Animal PhysiologyNeurotransmitter Receptor Influence on Behavior