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Design and synthesis of the first indole-based blockers of Panx-1 channel

Letizia Crocetti, Gabriella Guerrini, Sara Puglioli, Maria Paola Giovannoni, Lorenzo Di Cesare Mannelli, Elena Lucarini, Carla Ghelardini, Junjie Wang, Gerhard Dahl

2021European Journal of Medicinal Chemistry18 citationsDOIOpen Access PDF

Topics & Concepts

ChemistryIndole testIn vivoPharmacologyStereochemistryMedicineBiotechnologyBiologyIon channel regulation and functionNicotinic Acetylcholine Receptors StudyCardiac electrophysiology and arrhythmias
Design and synthesis of the first indole-based blockers of Panx-1 channel | Litcius